Vol. 3 No. 1 (2015) | ADMET and DMPK

Vol. 3 No. 1 (2015)

Transporters and permeability

Guest editor: Kiyohiko Sugano

Published: 03-04-2015

Reviews

The extended clearance model and its use for the interpretation of hepatobiliary elimination data

Gian Camenisch, Julia Riede, Annett Kunze, Jörg Huwyler, Birk Poller, Kenichi Umehara

ADMET and DMPK, Vol. 3 No. 1 (2015), 1-14

Published 31-03-2015;

DOI: https://doi.org/10.5599/admet.3.1.144
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Original Scientific Articles

Expression and Transport of a-Synuclein at the Blood-Cerebrospinal Fluid Barrier and Effects of Manganese Exposure

Christopher A Bates, Sherleen Fu, Daniel Ysselstein, Jean-Christophe Rochet, Wei Zheng

ADMET and DMPK, Vol. 3 No. 1 (2015), 15-33

Published 31-03-2015;

DOI: https://doi.org/10.5599/admet.3.1.159
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Characterization of SLC transporters in human skin

Marion Alriquet, Karine Sevin, Alexandre Gaborit, Pierre Comby, Bernard Ruty, Hanan Osman-Ponchet

ADMET and DMPK, Vol. 3 No. 1 (2015), 34-44

Published 31-03-2015;

DOI: https://doi.org/10.5599/admet.3.1.163
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Effect of Bioenhancers on Amoxicillin bioavailability

Kalyani Barve, Kushal Ruparel

ADMET and DMPK, Vol. 3 No. 1 (2015), 45-50

Published 31-03-2015;

DOI: https://doi.org/10.5599/admet.3.1.161
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Adaptation of a human gut epithelial model in relation to the assessment of clinical pharmacokinetic parameters for selected tyrosine kinase inhibitors

Richard Honeywell, Christien Fatmawati, Marita Buddha, Sarina Hitzerd, Ietje Kathman, Godefridus Peters

ADMET and DMPK, Vol. 3 No. 1 (2015), 51-67

Published 31-03-2015;

DOI: https://doi.org/10.5599/admet.3.1.169
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Short Communications

P-glycoprotein-dependent pharmacokinetics of irinotecan and its active metabolite, SN-38 in rats: Effect of verapamil

Tripta Garg, Manu Jaggi, Roop K. Khar, Sushama Talegaonkar

ADMET and DMPK, Vol. 3 No. 1 (2015), 68-76

Published 31-03-2015;

DOI: https://doi.org/10.5599/admet.3.1.154
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Notes

Differential effects of mitogen-activated protein kinase pathway inhibitors on P-glycoprotein activation

Hirokazu Wakuda, Shino Miyauchi, Kana Maruyama, Satomi Kagota, Kazuki Nakamura, Keizo Umegaki, Shizuo Yamada, Kazumasa Shinozuka

ADMET and DMPK, Vol. 3 No. 1 (2015), 77-83

Published 31-03-2015;

DOI: https://doi.org/10.5599/admet.3.1.142
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